Caralluma fimbriata is an important medicinal succulent plant traditionally used in India as a famine food and appetite suppressant. In recent years, scientific studies have shown that the plant possesses several pharmacological activities such as anti-obesity, antioxidant, antimicrobial, anti-inflammatory, antidiabetic, hypolipidemic and anticancer effects. These activities are mainly due to the presence of bioactive compounds like pregnane glycosides, flavonoids, phenols, tannins and saponins. Various in-vitro, in-vivo and clinical studies have demonstrated its therapeutic potential with minimal adverse effects. This review summarizes the phytochemistry, traditional uses, pharmacological activities and future therapeutic importance of Caralluma fimbriata.
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